SCHEMBL4748788

SCHEMBL4748788

O=C(C=Cc1ccc(Cl)cc1)c1cccc(Nc2ccnc3cc(Cl)ccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.52
CYP1A2 P05177 4/20 0.52
MAPT P10636 4/20 0.51
GAA P10253 2/20 0.51
ATM Q13315 1/20 0.51
PTGS2 P35354 2/20 0.51
MET P08581 1/20 0.51
APP P05067 2/20 0.49
NR4A2 P43354 2/20 0.49
FADS1 O60427 1/20 0.49
DNMT1 P26358 1/20 0.47
DNMT3A Q9Y6K1 1/20 0.47
ABCB1 P08183 3/20 0.47
ABCG2 Q9UNQ0 3/20 0.47
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KCNH2 Q12809 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14024396 1.00 CYP2D6 (0.52) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL4748773 0.95 GAA (0.59) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL4748784 0.90 CYP2D6 (0.52) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL14024471 0.90 APP (0.46) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL14024382 0.89 MAPT (0.60) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL4748932 0.89 MAPT (0.60) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL4748929 0.89 MAPT (0.60) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL14024410 0.85 GAA (0.59) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL30383538 0.85 GAA (0.59) CYP2D6CYP1A2MAPTGAAATM
SCHEMBL4748776 0.83 GAA (0.56) CYP2D6CYP1A2MAPTGAAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed