SCHEMBL4748908

SCHEMBL4748908

CO[C@H]1CN(C)CCc2sc(Br)cc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 7/20 0.33
DRD5 P21918 4/20 0.33
CYP2D6 P10635 2/20 0.32
CYP3A4 P08684 1/20 0.32
DRD2 P14416 2/20 0.31
CYP1A2 P05177 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ADCY2 Q08462 1/20 0.31
LMNA P02545 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
SLC6A2 P23975 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
MAPK1 P28482 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3308477 1.00 DRD1 (0.33) DRD1DRD5CYP2D6CYP3A4DRD2
SCHEMBL4752668 0.84 NPC1 (0.32)
SCHEMBL4748999 0.80 DRD1 (0.35) DRD1DRD5CYP2D6DRD2CYP1A2
SCHEMBL4752664 0.79 ALDH1A1 (0.37) DRD1CYP2D6CYP3A4HSD17B10SLC6A2
SCHEMBL3310259 0.79 ALDH1A1 (0.37) DRD1CYP2D6CYP3A4HSD17B10SLC6A2
SCHEMBL3307455 0.78 HPGD (0.40) CYP1A2HSD17B10LMNASLC6A2MAPK1
SCHEMBL4751943 0.78 DRD1 (0.34) DRD1DRD5CYP2D6CYP3A4DRD2
SCHEMBL4435809 0.77 SLC6A2 (0.32) CYP2D6CYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL4431719 0.76 SLC6A2 (0.31) SLC6A2SLC6A4SLC6A3ALOX15
SCHEMBL3002089 0.75 POLB (0.40) CYP2C19HSD17B10LMNAMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135526-A1 CARBOXYLIC ACID AMIDES AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO disclosed