SCHEMBL4748942

SCHEMBL4748942

O=C1CN(Cc2ccc(F)cc2)CCN1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
POLB P06746 1/20 0.61
GRM2 Q14416 1/20 0.54
MCHR1 Q99705 2/20 0.48
KMT2A Q03164 3/20 0.44
ATM Q13315 1/20 0.44
KDM4E B2RXH2 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
MEN1 O00255 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
ADRA2C P18825 1/20 0.42
CCR2 P41597 1/20 0.42
CXCL12 P48061 1/20 0.42
BLM P54132 1/20 0.42
CXCR4 P61073 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751222 0.85 SMN1; SMN2 (0.58) ALDH1A1POLBKMT2AATMKDM4E
SCHEMBL990427 0.84 KCNH2 (0.50) ALDH1A1POLBGRM2MCHR1
SCHEMBL3149433 0.84 ALDH1A1 (0.50) ALDH1A1POLBGRM2KMT2AATM
SCHEMBL17468364 0.84 CXCR4 (0.55) ALDH1A1POLBKMT2AATMKDM4E
SCHEMBL1427302 0.84 ALDH1A1 (0.47) ALDH1A1POLBKMT2AATMKDM4E
SCHEMBL220097 0.83 SIGMAR1 (0.62) ALDH1A1KMT2AATMSMN1; SMN2MEN1
SCHEMBL21133116 0.83 ALDH1A1 (0.53) ALDH1A1POLBGRM2MCHR1KMT2A
SCHEMBL14045873 0.83 CXCR4 (0.55) ALDH1A1POLBGRM2MCHR1KMT2A
SCHEMBL6707988 0.81 KMT2A (0.43) ALDH1A1POLBGRM2KMT2AATM
SCHEMBL27713409 0.80 ALDH1A1 (0.53) ALDH1A1POLBGRM2KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008136754-A1 NOVEL BENZYL - 2 -OXO-PIPERAZINYL/ 7-OXO/5-OXA- [1,4] DIAZEPANYL/ 2 -OXO- TETRAHYDROPYRIMIDINYL DERIVATIVES ASTRAZENECA AB (SE) 2008-11-13 WO claimed
WO-2008136754-A1 NOVEL BENZYL - 2 -OXO-PIPERAZINYL/ 7-OXO/5-OXA- [1,4] DIAZEPANYL/ 2 -OXO- TETRAHYDROPYRIMIDINYL DERIVATIVES ASTRAZENECA AB (SE) 2008-11-13 WO disclosed