SCHEMBL4749634

SCHEMBL4749634

Cc1ccc([N+](=O)[O-])c(NC2CCN(C(=O)O)CC2C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 2/20 0.42
MCOLN3 Q8TDD5 1/20 0.40
NPC1 O15118 1/20 0.39
MAPT P10636 5/20 0.39
MAPK1 P28482 2/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPBWR1 P48145 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MCHR1 Q99705 1/20 0.37
KAT2B Q92831 1/20 0.37
HTT P42858 2/20 0.37
DCTPP1 Q9H773 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749628 1.00 GRK6 (0.42) GRK6MCOLN3NPC1MAPTMAPK1
SCHEMBL14041860 0.87 LMNA (0.46) GRK6NPC1MAPTMAPK1ALDH1A1
SCHEMBL30960353 0.83 APP (0.44) NPC1MAPTMAPK1ALDH1A1KDM4E
SCHEMBL4746315 0.82 TP53 (0.37) NPC1MEN1KMT2ASMN1; SMN2CYP2C9
SCHEMBL11909744 0.78 KAT2B (0.45) GRK6MCOLN3MAPTMAPK1ALDH1A1
SCHEMBL11909741 0.78 KAT2B (0.45) GRK6MCOLN3MAPTMAPK1ALDH1A1
SCHEMBL11272299 0.76 MAPT (0.47) NPC1MAPTMAPK1ALDH1A1MEN1
SCHEMBL11272273 0.76 MAPT (0.47) NPC1MAPTMAPK1ALDH1A1MEN1
SCHEMBL11836392 0.74 PKM (0.45) NPC1MAPTMAPK1ALDH1A1KDM4E
SCHEMBL4749021 0.74 MAPT (0.44) GRK6MCOLN3NPC1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008119718-A1 COMPOUNDS WHICH HAVE ACTIVITY AT M1 RECEPTOR AND THEIR USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2008-10-09 WO disclosed