SCHEMBL4750064

SCHEMBL4750064

O=C(O)N1CCNC(CCOc2cc(F)cc(F)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA4 P22748 4/20 0.36
CA9 Q16790 4/20 0.36
CCR3 P51677 1/20 0.34
PARP1 P09874 1/20 0.34
SCN9A Q15858 6/20 0.33
REN P00797 1/20 0.33
SOD1 P00441 1/20 0.33
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291240 1.00 CA1 (0.36) CA1CA2CA4CA9CCR3
SCHEMBL4291606 0.90 SCN9A (0.38) SCN9A
SCHEMBL4292524 0.88 LTA4H (0.39) CCR3PARP1SCN9A
SCHEMBL4284889 0.85 SCN9A (0.40) SCN9ASOD1
SCHEMBL3493396 0.84 TEAD1 (0.46) CA1CA2CA4CA9PARP1
SCHEMBL8118778 0.83 CXCR4 (0.43)
Hydrochloric Acid SCHEMBL4293711 0.82 PARP1 (0.45) CA1CA2CA4CA9PARP1
Hydrochloric Acid SCHEMBL4293709 0.82 PARP1 (0.45) CA1CA2CA4CA9PARP1
SCHEMBL4282373 0.81 L3MBTL1 (0.47) CA1CA2CA4CA9PARP1
SCHEMBL4751897 0.81 L3MBTL1 (0.47) CA1CA2CA4CA9PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed