SCHEMBL4750144

SCHEMBL4750144

Nc1ccc(NC(=O)CCC2CCNC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LDLR P01130 1/20 0.47
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
ROCK2 O75116 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746331 0.85 HDAC3 (0.54) LDLRITGB3ITGA2BROCK2HDAC3
SCHEMBL29223347 0.79 KLK7 (0.57) ITGB3ITGA2BHDAC3HDAC1HDAC2
SCHEMBL6508976 0.78 KMT2A (0.67) ROCK2KMT2AALDH1A1NPSR1
SCHEMBL10198173 0.77 ROCK2 (0.61) LDLRROCK2KMT2AALDH1A1
SCHEMBL31227621 0.76 KMT2A (0.60) ROCK2HDAC3HDAC1HDAC2KMT2A
SCHEMBL15197080 0.75 MAPT (0.64) HDAC3HDAC1HDAC2KMT2A
SCHEMBL28051643 0.74
SCHEMBL29690252 0.74 NPSR1 (0.50) LDLRITGB3ITGA2BROCK2HDAC3
Hydrochloric Acid SCHEMBL28051567 0.73
SCHEMBL29850847 0.72 EPHX2 (0.63) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008122667-A2 UREYLENE DERIVATIVES SCHOOL OF PHARMACY (GB) 2008-10-16 WO disclosed