SCHEMBL4750177

SCHEMBL4750177

O=C(O)N1CCNC(Cc2ccc(Cl)cc2Cl)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.43
CYP3A4 P08684 2/20 0.43
UGCG Q16739 2/20 0.43
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
CA9 Q16790 2/20 0.39
FFAR1 O14842 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2J2 P51589 1/20 0.39
KMT2A Q03164 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
S1PR1 P21453 1/20 0.38
LTK P29376 1/20 0.38
TAOK1 Q7L7X3 1/20 0.38
S1PR5 Q9H228 1/20 0.38
MC4R P32245 2/20 0.38
MC5R P33032 2/20 0.38
MC3R P41968 2/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4282776 1.00 EPHX2 (0.43) EPHX2CYP3A4UGCGCA1CA2
SCHEMBL13705075 0.83 ALDH1A1 (0.48) CYP3A4UGCGKMT2A
SCHEMBL4749948 0.74 CA1 (0.62) CA1CA2CA4CA9KMT2A
SCHEMBL5719329 0.74 CA1 (0.62) CA1CA2CA4CA9KMT2A
SCHEMBL3495230 0.74 CA1 (0.62) CA1CA2CA4CA9KMT2A
SCHEMBL3492392 0.72 CA1 (0.51) CA1CA2CA4CA9CCR3
SCHEMBL2578568 0.71 NPC1 (0.39) CA1CA2CA9KMT2AHPGD
SCHEMBL4286365 0.71 PTGDR2 (0.39) FFAR1KMT2AHPGD
SCHEMBL4290915 0.71 KMT2A (0.41) KMT2A
SCHEMBL4281831 0.71 RAB9A (0.40) CYP3A4KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed