SCHEMBL4750823

SCHEMBL4750823

O=C1[N]c2cccc(F)c2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 3/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA4 P22748 1/20 0.40
PARP1 P09874 3/20 0.39
HTR5A P47898 1/20 0.36
PDE7A Q13946 1/20 0.36
AKR1B1 P15121 1/20 0.33
AR P10275 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
DAO P14920 3/20 0.33
DDO Q99489 1/20 0.33
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
TYMS P04818 1/20 0.31
IKBKB O14920 1/20 0.31
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4753125 0.76 CA9 (0.40) CA9CA12CA1CA2CA7
SCHEMBL4753134 0.76 CES1 (0.44) CA9CA12CA1CA2CA7
SCHEMBL4752983 0.68 PARP1 (0.37) CA9CA12CA1CA2CA7
SCHEMBL20505096 0.66 MAPT (0.44)
SCHEMBL20723 0.66 MAPT (0.44)
SCHEMBL2165115 0.65 CA12 (0.42) CA9CA12CA1CA2CA7
SCHEMBL3826696 0.63 GRM5 (0.30)
SCHEMBL21296775 0.63 GSK3B (0.52) CA9CA12CA1CA2CA7
SCHEMBL555451 0.63 GSK3B (0.52) CA9CA12CA1CA2CA7
SCHEMBL1346633 0.62 CREBBP (0.39) CA9CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed