SCHEMBL4751007

SCHEMBL4751007

COc1ccc(Cn2nncc2C[AsH2])cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.46
NPBWR1 P48145 6/20 0.45
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
CMA1 P23946 1/20 0.42
MCHR1 Q99705 1/20 0.41
CYP19A1 P11511 1/20 0.41
HSD11B1 P28845 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PKM P14618 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MET P08581 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13151306 0.86 TOP2A (0.47) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL1031479 0.85 TOP2A (0.49) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL19631128 0.82 TAAR1 (0.51) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL31284789 0.81 TOP2A (0.48) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL30946374 0.80 TOP2A (0.52) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL18377688 0.80 ALDH1A1 (0.54) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL31285046 0.78 TOP2A (0.48) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL13151274 0.77 NPBWR1 (0.46) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL18367564 0.76 TOP2A (0.49) TOP2ANPBWR1ALDH1A1KDM4EMAPT
SCHEMBL27840090 0.75 TOP2A (0.48) TOP2ANPBWR1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904489-A2 PROCESS FOR THE SYNTHESIS OF TRIAZOLES Rib-X Pharmaceuticals, Inc. (US) 2008-04-02 EP disclosed
WO-2006133397-A2 PROCESS FOR THE SYNTHESIS OF TRIAZOLES RIB-X PHARMACEUTICALS, INC. (US) 2006-12-14 WO disclosed