SCHEMBL4751305

SCHEMBL4751305

Fc1ccc(OCCC2CCN(Cc3nc4cccc5c4n3CCO5)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A2 P23975 1/20 0.38
LIPG Q9Y5X9 1/20 0.38
CHRM4 P08173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4945433 0.92 DRD2 (0.36) SLC6A3SLC6A4SLC6A2LIPGCHRM4
SCHEMBL4751794 0.90 GRM2 (0.38) LIPG
SCHEMBL4693428 0.87 CHEK2 (0.38) SLC6A3SLC6A4SLC6A2
SCHEMBL4745230 0.86 MAOB (0.43) SLC6A3SLC6A4LIPG
SCHEMBL4947552 0.84 CYP2D6 (0.39) SLC6A3SLC6A4LIPG
SCHEMBL4950186 0.83 NPC1 (0.43) SLC6A3SLC6A4SLC6A2CHRM4
SCHEMBL13993059 0.82 DRD2 (0.43) CHRM4
SCHEMBL4146888 0.79 NPY1R (0.41)
SCHEMBL4750532 0.77 GRM2 (0.45) SLC6A4
SCHEMBL4941482 0.76 LIPG (0.36) LIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080318999-A1 Tricyclic Benzimidazoles and Their Use as Metabotropic Glutamate Receptor Modulators ASTRAZENECA AB (SE) 2008-12-25 US claimed
EP-1912989-A2 TRICYCLIC BENZIMIDAZOLES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-04-23 EP claimed
WO-2007018998-A2 TRICYCLIC BENZIMIDAZOLES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-02-15 WO claimed
US-20070032469-A1 Tricyclic benzimidazoles and their use as metabotropic glutamate receptor modulators ASTRAZENECA AB (SE) 2007-02-08 US claimed
CN-115485431-A Treating agent for synthetic fiber, and method for treating synthetic fiber 竹本油脂株式会社 2022-12-16 CN disclosed
CN-111764173-A Treating agent for elastic fiber and elastic fiber 竹本油脂株式会社 2020-10-13 CN disclosed
US-20080318999-A1 Tricyclic Benzimidazoles and Their Use as Metabotropic Glutamate Receptor Modulators ASTRAZENECA AB (SE) 2008-12-25 US disclosed
US-20080318999-A1 Tricyclic Benzimidazoles and Their Use as Metabotropic Glutamate Receptor Modulators ASTRAZENECA AB (SE) 2008-12-25 US disclosed
US-20070042916-A1 METHODS FOR IMPROVED POWER TRANSMISSION PERFORMANCE AND COMPOSITIONS THEREFOR AFTON CHEMICAL CORPORATION 2007-02-22 US disclosed
WO-2007018998-A2 TRICYCLIC BENZIMIDAZOLES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-02-15 WO disclosed
US-20070032469-A1 Tricyclic benzimidazoles and their use as metabotropic glutamate receptor modulators ASTRAZENECA AB (SE) 2007-02-08 US disclosed
US-20070032469-A1 Tricyclic benzimidazoles and their use as metabotropic glutamate receptor modulators ASTRAZENECA AB (SE) 2007-02-08 US disclosed
US-20070000745-A1 METHODS FOR IMPROVED POWER TRANSMISSION PERFORMANCE AFTON CHEMICAL CORPORATION 2007-01-04 US disclosed
US-20070004603-A1 METHODS FOR IMPROVED POWER TRANSMISSION PERFORMANCE AND COMPOSITIONS THEREFOR AFTON CHEMICAL CORPORATION 2007-01-04 US disclosed
EP-1739158-A2 Methods for improved power transmission performance and lubricating compositions therefor Afton Chemical Corporation (US) 2007-01-03 EP disclosed
EP-1739321-A2 Methods for improved power transmission performance Afton Chemical Corporation (US) 2007-01-03 EP disclosed
EP-1739159-A2 Methods for improved power transmission performance and lubricating compositions therefor Afton Chemical Corporation (US) 2007-01-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032469-A1 Tricyclic benzimidazoles and their use as metabotropic glutamate receptor modulators GRM2, GRM1, GRIN2B SLC6A3 122/4885SLC6A4 115/4885SLC6A2 143/4885
US-20080318999-A1 Tricyclic Benzimidazoles and Their Use as Metabotropic Glutamate Receptor Modulators GRM2, GRM1, GRIN2B SLC6A3 122/4885SLC6A4 115/4885SLC6A2 143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.