SCHEMBL4751330

SCHEMBL4751330

O=Cc1ccccc1-c1cccc(Nc2ccnc3cc(Cl)ccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 1/20 0.54
APP P05067 2/20 0.51
NR4A2 P43354 2/20 0.51
MAPT P10636 5/20 0.50
GAA P10253 2/20 0.50
ATM Q13315 1/20 0.50
ALK Q9UM73 1/20 0.49
CYP1A2 P05177 6/20 0.48
CYP2D6 P10635 6/20 0.48
CA9 Q16790 1/20 0.48
KDR P35968 2/20 0.48
EGFR P00533 2/20 0.48
AURKA O14965 1/20 0.48
INSR P06213 1/20 0.48
IGF1R P08069 1/20 0.48
SRC P12931 1/20 0.48
EPHB4 P54760 1/20 0.48
TEK Q02763 1/20 0.48
AURKB Q96GD4 1/20 0.48
POLB P06746 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751312 0.83 POLB (0.55) NR4A2MAPTGAAATMCYP1A2
Metaquine SCHEMBL7205743 0.80 FADS1 (0.71) FADS1APPNR4A2MAPTGAA
SCHEMBL5309628 0.77 MAPT (0.74) FADS1APPNR4A2MAPTGAA
SCHEMBL29950963 0.77 GAA (0.65) APPNR4A2MAPTGAAATM
SCHEMBL5591942 0.76 GRM4 (0.47) NR4A2MAPTCYP1A2POLBKMT2A
SCHEMBL9482173 0.74 MAPT (0.69) APPNR4A2MAPTGAAATM
SCHEMBL2011565 0.74 GAA (0.73) FADS1APPNR4A2MAPTGAA
SCHEMBL30179800 0.74 GAA (0.73) FADS1APPNR4A2MAPTGAA
SCHEMBL19633680 0.74 FADS1 (0.63) FADS1APPNR4A2MAPTGAA
SCHEMBL5257871 0.74 KDR (0.81) FADS1APPNR4A2MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed