SCHEMBL4752370

SCHEMBL4752370

Cc1cnc(Br)nc1Br

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27980126 0.79
SCHEMBL12352066 0.79
SCHEMBL26658795 0.75
SCHEMBL21737363 0.75
SCHEMBL29144926 0.75
SCHEMBL24225498 0.72 NUDT1 (0.34)
SCHEMBL25928370 0.72 APLNR (0.33)
SCHEMBL26860463 0.72 HPGD (0.33)
SCHEMBL26860462 0.72 TDP1 (0.31)
SCHEMBL25928373 0.72 CCR1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025264278-A1 ERK2 DEGRADERS MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2025-12-26 WO disclosed
WO-2024233665-A1 COMPOUNDS AND THEIR USE AGAINST CANCER TANGO THERAPEUTICS, INC. (US) 2024-11-14 WO disclosed
US-20230159508-A1 INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2023-05-25 US disclosed
US-9422271-B2 Pyrimidine compounds as tuberculosis inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-08-23 US disclosed
US-20140249137-A1 PYRIMIDINE COMPOUNDS AS TUBERCULOSIS INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-09-04 US disclosed
US-20110053916-A1 PYRIMIDINE COMPOUNDS AS TUBERCULOSIS INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-03 US disclosed
WO-2008147831-A1 ANTHRANILAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2008-12-04 WO disclosed
WO-2008147831-A1 ANTHRANILAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2008-12-04 WO disclosed