SCHEMBL4752422

SCHEMBL4752422

O=C1[N]c2cc(Cl)ccc2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.44
TGM2 P21980 2/20 0.44
PPOX P50336 1/20 0.44
AHR P35869 2/20 0.43
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CMA1 P23946 1/20 0.39
CHEK1 O14757 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
TSHR P16473 1/20 0.38
ABCC8 Q09428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817144 1.00 CES1 (0.44) CES1TGM2PPOXAHRCA12
SCHEMBL2719976 0.84 CES1 (0.44) CES1TGM2PPOXAHRCA12
SCHEMBL4753132 0.76 TGM2 (0.44) CES1TGM2AHRCA12CA1
SCHEMBL4382993 0.76 TGM2 (0.44) CES1TGM2CYP1A2CYP3A4CYP2D6
SCHEMBL6264592 0.76 CA1 (0.40) CA12CA1CA2CA4CA7
SCHEMBL1401519 0.76 ROS1 (0.41) CA12CA1CA2CA4CA7
SCHEMBL1695075 0.76 CA9 (0.38) CA12CA9CYP3A4ALDH1A1TSHR
SCHEMBL4750469 0.76 CA1 (0.40) CA12CA1CA2CA4CA7
SCHEMBL473854 0.76 TGM2 (0.44) CES1TGM2AHRCA12CA1
SCHEMBL6219325 0.75 CES1 (0.41) CES1CYP1A2CYP3A4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed