SCHEMBL4750469

SCHEMBL4750469

O=C1[N]c2cc(F)ccc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA12 O43570 1/20 0.40
CA4 P22748 1/20 0.40
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRM1 P11229 1/20 0.37
HRH1 P35367 1/20 0.37
PAK1 Q13153 1/20 0.37
HTR5A P47898 2/20 0.36
GRM5 P41594 2/20 0.36
KDM4E B2RXH2 1/20 0.35
NOX1 Q9Y5S8 1/20 0.34
AKR1B1 P15121 3/20 0.33
LRRK2 Q5S007 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6264592 1.00 CA1 (0.40) CA1CA2CA7CA9CA12
SCHEMBL4750491 0.84 HTR5A (0.36) CA1CA2CA7CA9CA12
SCHEMBL8555842 0.81 KMT2A (0.39) CA1CA2CA7CA9CA12
SCHEMBL6222347 0.77 KIF11 (0.41) KMT2AKDM4EPARP1
SCHEMBL7514332 0.77 LRRK2 (0.41) CA1CA2CA7CA9CA12
SCHEMBL473854 0.76 TGM2 (0.44) CA1CA2CA7CA9CA12
SCHEMBL1695075 0.76 CA9 (0.38) CA9CA12MAPTKMT2AKDM4E
SCHEMBL1401519 0.76 ROS1 (0.41) CA1CA2CA7CA9CA12
SCHEMBL4382993 0.76 TGM2 (0.44) CYP1A2MAPTCYP2C19KMT2ALRRK2
SCHEMBL4752422 0.76 CES1 (0.44) CA1CA2CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed