SCHEMBL4752467

SCHEMBL4752467

O=C1[N]c2c(cccc2C(F)(F)F)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.41
PARP1 P09874 1/20 0.38
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HSD17B10 Q99714 1/20 0.37
AXL P30530 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
NOTUM Q6P988 3/20 0.34
AR P10275 1/20 0.34
PDE7A Q13946 1/20 0.34
APAF1 O14727 1/20 0.33
USP2 O75604 1/20 0.33
PLCG1 P19174 1/20 0.33
CCR6 P51684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587215 0.76 PLAUR (0.31)
SCHEMBL4752983 0.76 PARP1 (0.37) PARP1AR
SCHEMBL6120237 0.72 PARP1 (0.33) PARP1HSD17B10ALDH1A1MEN1POLB
SCHEMBL4750499 0.72 CES1 (0.44) CES1PARP1PDE7A
SCHEMBL6230711 0.72 MEN1 (0.37) PARP1KDM4ESMN1; SMN2HSD17B10ALDH1A1
SCHEMBL5132320 0.68 TDP1 (0.44) PARP1KDM4ESMN1; SMN2HSD17B10ALDH1A1
SCHEMBL1451647 0.66 CES1 (0.42) CES1PARP1KDM4ESMN1; SMN2HSD17B10
SCHEMBL6179037 0.66 CES1 (0.55) CES1PARP1KDM4ESMN1; SMN2HSD17B10
SCHEMBL3741907 0.65
SCHEMBL17974653 0.64 AHR (0.44) CES1KDM4EMEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008146064-A1 NEW BENZOFURAN DERIVATIVES AS SELECTIVE 5HT7 RECEPTOR INHIBITORS AND PROCESS FOR THEIR PREPARATION EGIS GYÓGYSZERGYÁR (HU) 2008-12-04 WO disclosed