SCHEMBL4752483

SCHEMBL4752483

O=C(O)N1CCNC(CCOc2c(F)cccc2F)C1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
REN P00797 7/20 0.38
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA4 P22748 4/20 0.38
CA9 Q16790 4/20 0.38
PARP1 P09874 2/20 0.35
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
ATM Q13315 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSP90AA1 P07900 1/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCR3 P51677 1/20 0.34
NTRK1 P04629 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4281538 1.00 REN (0.38) RENCA1CA2CA4CA9
Hydrochloric Acid SCHEMBL4290984 0.90 SCN9A (0.38) RENRAB9AKDM4EALDH1A1CCR3
SCHEMBL4287415 0.88 REN (0.39) RENCA1CA2CA4CA9
Hydrochloric Acid SCHEMBL4281883 0.86 NPC1 (0.43) CA1CA2CA4CA9RAB9A
SCHEMBL8126494 0.85 CXCR4 (0.45) CA1CA2CA4CA9RAB9A
SCHEMBL3493396 0.83 TEAD1 (0.46) RENCA1CA2CA4CA9
SCHEMBL4290277 0.82 CCR3 (0.39) RENCA1CA2CA4CA9
SCHEMBL4752929 0.82 CCR3 (0.39) RENCA1CA2CA4CA9
Hydrochloric Acid SCHEMBL4293711 0.81 PARP1 (0.45) RENCA1CA2CA4CA9
Hydrochloric Acid SCHEMBL4293709 0.81 PARP1 (0.45) RENCA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed