SCHEMBL4752839

SCHEMBL4752839

Cc1c(F)cccc1C1C(C(=O)c2cccc(O)c2)CN(CCCCNC2CCC2)CC1C(=O)C1CN(CCCCNC2CCC2)CC(C(=O)c2cccc(O)c2)C1c1cccc(F)c1C

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.34
DRD2 P14416 2/20 0.34
HTR1A P08908 2/20 0.34
DRD1 P21728 2/20 0.34
DRD4 P21917 2/20 0.34
DRD5 P21918 2/20 0.34
GRM5 P41594 2/20 0.32
KDM2B Q8NHM5 3/20 0.31
OPRL1 P41146 1/20 0.31
ADRA1A P35348 1/20 0.31
MCHR1 Q99705 1/20 0.31
KMT2A Q03164 1/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752837 1.00 DRD3 (0.34) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749235 0.97 DRD3 (0.35) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749218 0.97 DRD3 (0.35) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749510 0.89 DRD3 (0.34) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749471 0.89 DRD3 (0.34) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4751841 0.87 DRD3 (0.34) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4751833 0.87 DRD3 (0.34) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749105 0.87 MET (0.36) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4749501 0.87 DRD3 (0.33) DRD3DRD2HTR1ADRD1DRD4
SCHEMBL4752868 0.87 DRD2 (0.33) DRD3DRD2HTR1ADRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO claimed
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed