SCHEMBL4753396

SCHEMBL4753396

O=C(O)N1CCNC(CCn2cc3ccccc3n2)C1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA4 P22748 4/20 0.36
CA9 Q16790 4/20 0.36
LCK P06239 1/20 0.35
MCHR1 Q99705 2/20 0.34
PARP1 P09874 2/20 0.34
ADRB1 P08588 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
REN P00797 3/20 0.33
KDM5A P29375 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
SCN9A Q15858 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4286425 1.00 CA1 (0.36) CA1CA2CA4CA9LCK
SCHEMBL4285115 0.94 CA1 (0.35) CA1CA2CA4CA9LCK
SCHEMBL13705142 0.86 GRIN2B (0.43) CA1CA2CA4CA9LCK
SCHEMBL13705147 0.80 GRIN2B (0.44) PARP1
SCHEMBL4284114 0.79 MCHR1 (0.35) CA1CA2CA4CA9MCHR1
SCHEMBL4282685 0.78 PDE10A (0.40) CA1CA2CA4CA9PARP1
SCHEMBL4290999 0.76 KMO (0.50) CA1CA2CA4CA9REN
SCHEMBL4287498 0.76 EGLN3 (0.50)
SCHEMBL4290072 0.76 EGLN3 (0.50) LCK
SCHEMBL4753442 0.76 KMO (0.50) CA1CA2CA4CA9REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed