SCHEMBL4753472

SCHEMBL4753472

O=CC(NCc1ccc(-c2ccccc2)cc1)N1CCN(C(=O)c2cc(F)ccc2C(F)(F)F)CC1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 7/20 0.47
SCN9A Q15858 7/20 0.47
SMO Q99835 1/20 0.41
SCD O00767 2/20 0.40
DCTPP1 Q9H773 1/20 0.39
EPHX2 P34913 1/20 0.38
MAPK8 P45983 2/20 0.38
MAPK10 P53779 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2B P41595 1/20 0.38
MAPK14 Q16539 1/20 0.38
PPARG P37231 2/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4753878 0.90 CYP2C9 (0.47) SCDDCTPP1MAPK8MAPK10CYP2C9
SCHEMBL4753491 0.89 SCN5A (0.38) SCN5ASCN9ASMOSCDEPHX2
Hydrochloric Acid SCHEMBL3467141 0.88 SCN5A (0.38) SCN5ASCN9ASMOSCDEPHX2
SCHEMBL4753766 0.85 SCD5 (0.42) SCN5ASCN9ASCDEPHX2
SCHEMBL1221107 0.82 SCN5A (0.44) SCN5ASCN9ASMOSCDDCTPP1
SCHEMBL3466775 0.79 SCN5A (0.46) SCN5ASCN9AHTR2B
Hydrochloric Acid SCHEMBL3466605 0.79 SCN5A (0.45) SCN5ASCN9AHTR2B
Hydrochloric Acid SCHEMBL4755658 0.77 SMO (0.43) SCN5ASCN9ASMOSCDCYP2C9
SCHEMBL13059058 0.76 SMO (0.44) SCN5ASCN9ASMOSCDPPARG
Hydrochloric Acid SCHEMBL4755567 0.76 SCD (0.44) SMOSCDDCTPP1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157844-A1 NOVEL PIPERAZINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-12-24 WO disclosed