SCHEMBL4753765

SCHEMBL4753765

NC(C=O)N1CCN(C(=O)c2cc(F)ccc2C(F)(F)F)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
SCD O00767 1/20 0.43
P2RX7 Q99572 5/20 0.39
HDAC8 Q9BY41 1/20 0.39
SCN5A Q14524 2/20 0.39
SCN9A Q15858 2/20 0.39
MGLL Q99685 1/20 0.39
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
SLC9A1 P19634 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3466376 0.99 HCRTR1 (0.43) HCRTR1HCRTR2SCDP2RX7HDAC8
SCHEMBL4753470 0.84 SCD (0.51) SCDP2RX7MGLLCYP2C9CYP2C19
Hydrochloric Acid SCHEMBL3466569 0.83 SCD (0.50) SCDP2RX7MGLLCYP2C9CYP2C19
SCHEMBL4772658 0.82 CACNA2D1 (0.39) HCRTR1HCRTR2SCDP2RX7SCN5A
Hydrochloric Acid SCHEMBL3466281 0.82 SCN5A (0.51) SCDP2RX7HDAC8SCN5ASCN9A
SCHEMBL4775889 0.81 SCN5A (0.42) HCRTR1HCRTR2SCDP2RX7HDAC8
SCHEMBL4774662 0.80 CACNA1B (0.41) HCRTR1HCRTR2SCDHDAC8SCN5A
Hydrochloric Acid SCHEMBL3468340 0.79 RBP4 (0.53) SCDPSEN1PSEN2APH1BNCSTN
SCHEMBL4837579 0.79 SCD (0.38) HCRTR1HCRTR2SCDP2RX7HDAC8
SCHEMBL2820773 0.79 HCRTR1 (0.48) HCRTR1HCRTR2SCDP2RX7MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157844-A1 NOVEL PIPERAZINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-12-24 WO disclosed