SCHEMBL4753872

SCHEMBL4753872

CN(CCN(CCCN)c1cccc(Cl)c1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
KDM4E B2RXH2 2/20 0.42
AOC3 Q16853 1/20 0.42
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
ADRA2C P18825 1/20 0.39
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
SLC6A7 Q99884 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
CCR5 P51681 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499700 0.83 MAPT (0.44) MAPTKDM4EAOC3HTR3EHTR3B
SCHEMBL4753581 0.81 TMEM97 (0.45) MAPTKDM4ETMEM97SIGMAR1ALDH1A1
SCHEMBL11133767 0.71 MAPT (0.65) MAPTKDM4EAOC3HTR3EHTR3B
SCHEMBL18300919 0.69 CRHBP (0.52) AOC3ALDH1A1RAB9AMEN1KMT2A
SCHEMBL2096198 0.69 HTR3E (0.61) MAPTKDM4EHTR3EHTR3BHTR3A
SCHEMBL31715773 0.69 HTR3E (0.61) MAPTKDM4EHTR3EHTR3BHTR3A
SCHEMBL1937726 0.68
SCHEMBL11793760 0.68 TAAR1 (0.44) MAPTADRA2CSIGMAR1ALDH1A1HTT
SCHEMBL342097 0.68 MAPT (0.55) MAPTHTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL8378174 0.68 MAPT (0.48) MAPTKDM4EHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed