SCHEMBL4755161

SCHEMBL4755161

CN1CC2CCN(c3ccc(N4CCN(c5ccc(Cl)nn5)CC4)cc3)C2C1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.54
KCNH2 Q12809 2/20 0.48
CHRNB2 P17787 2/20 0.44
CHRNB4 P30926 2/20 0.44
CHRNA3 P32297 2/20 0.44
CHRNA4 P43681 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3065520 1.00 HRH3 (0.54) HRH3KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL3067701 0.87 HRH3 (0.55) HRH3KCNH2
SCHEMBL31200556 0.85 HRH3 (0.50) HRH3KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL3058263 0.79 HRH3 (0.63) HRH3KCNH2
SCHEMBL3061109 0.79 HRH3 (0.61) HRH3KCNH2
SCHEMBL25437423 0.77 NLRP3 (0.50) HRH3CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL31200506 0.77 NLRP3 (0.50) HRH3CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL3063131 0.77 HRH3 (0.54) HRH3KCNH2
SCHEMBL4697400 0.77 HRH3 (0.54) HRH3KCNH2
SCHEMBL3062935 0.77 HRH3 (0.60) HRH3KCNH2CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001885-A2 OCTAHYDRO-PYRROLO[3,4-B]PYRROLE DERIVATIVES Abbott Laboratories (US) 2008-12-17 EP disclosed
WO-2007100990-A2 OCTAHYDRO-PYRROLO[3,4-B] PYRROLE DERIVATIVES AND THEIR USE AS HISTAMINE-3 RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2007-09-07 WO disclosed