SCHEMBL4756396

SCHEMBL4756396

Cc1ccc(O)c(C(=O)Nc2nc(S(C)(=O)=O)cs2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
ALDH1A1 P00352 3/20 0.50
HPGD P15428 3/20 0.50
GAA P10253 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
HTT P42858 1/20 0.50
HSD17B10 Q99714 1/20 0.50
RCE1 Q9Y256 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GRM5 P41594 1/20 0.49
STAT3 P40763 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PLAU P00749 2/20 0.45
F2 P00734 1/20 0.45
F10 P00742 1/20 0.45
PLAT P00750 1/20 0.45
P2RX1 P51575 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756405 0.90 NPC1 (0.50) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL4756398 0.87 SORT1 (0.50) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL4757291 0.86 NPC1 (0.49) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL12994116 0.86 KDM4E (0.48) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL4757362 0.84 SORT1 (0.47) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL703934 0.84 NPC1 (0.67) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL12974190 0.83 GCK (0.41) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL4930389 0.81 NPC1 (0.53) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL29682864 0.81 NPC1 (0.53) NPC1RAB9AALDH1A1HPGDGAA
SCHEMBL4757285 0.81 RAB9A (0.64) NPC1RAB9AALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11850237-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2023-12-26 US disclosed
US-11850237-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2023-12-26 US disclosed
EP-3895706-A1 THIAZOLINIDE COMPOUNDS FOR TREATING NON-INFLUENZA VIRAL INFECTIONS Romark Laboratories, L.C. (US) 2021-10-20 EP disclosed
US-20210177809-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2021-06-17 US disclosed
US-10912768-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2021-02-09 US disclosed
US-20190307730-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2019-10-10 US disclosed
US-10363243-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2019-07-30 US disclosed
US-20180078533-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2018-03-22 US disclosed
US-20180078533-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2018-03-22 US disclosed
US-9820975-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2017-11-21 US disclosed
US-9345690-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2016-05-24 US disclosed
US-20150250768-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2015-09-10 US disclosed
US-20150250768-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA ROMARK LABORATORIES L.C. (US) 2015-09-10 US disclosed
US-9023877-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2015-05-05 US disclosed
US-9023877-B2 Compounds and methods for treating influenza ROMARK LABORATORIES L.C. (US) 2015-05-05 US disclosed
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES, L.C. 2012-05-17 US disclosed
US-8124632-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES, L.C. (US) 2012-02-28 US disclosed
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES L.C. 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150250768-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-10912768-B2 Compounds and methods for treating influenza HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-20180078533-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-20210177809-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-20190307730-A1 COMPOUNDS AND METHODS FOR TREATING INFLUENZA HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-11850237-B2 Compounds and methods for treating influenza HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC NPC1 585/4885RAB9A 1694/4885ALDH1A1 1605/4885
US-10363243-B2 Compounds and methods for treating influenza HIF1AN, HAVCR2, NEU1 NPC1 473/4885RAB9A 1890/4885ALDH1A1 77/4885
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC NPC1 585/4885RAB9A 1694/4885ALDH1A1 1605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.