SCHEMBL4756906

SCHEMBL4756906

CCOC(=O)c1cc(Cl)cc(C2CCNC2)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HTR3A P46098 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755037 0.92 CA12 (0.42) SLC6A2SLC6A4SLC6A3CA12CA1
SCHEMBL231497 0.81 MAPT (0.48)
SCHEMBL31385899 0.80 CA12 (0.49) HTR3ACA12CA1CA2CA7
SCHEMBL31386022 0.80 CA12 (0.49) HTR3ACA12CA1CA2CA7
SCHEMBL13985025 0.80 HTR3A (0.50) HTR3A
SCHEMBL4755119 0.79 PDE4A (0.45) CA12CA1CA2CA7CA9
SCHEMBL18617801 0.76 HTR3A (0.51) SLC6A2SLC6A4SLC6A3HTR3A
Oxalic Acid SCHEMBL829222 0.75 HTR3A (0.54) HTR3A
SCHEMBL7589274 0.74 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL2662880 0.74 CA12 (0.62) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed