SCHEMBL4757086

SCHEMBL4757086

CC(C)Oc1ccc2c(Cl)nc(C(=O)N3CCCC3C(=O)O)c(O)c2c1I

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
KMT2A Q03164 1/20 0.35
ACE P12821 5/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OGFRL1 Q5TC84 1/20 0.34
REN P00797 2/20 0.34
KDM4E B2RXH2 1/20 0.34
F2 P00734 1/20 0.34
LMNA P02545 1/20 0.34
LTA4H P09960 1/20 0.34
MAPT P10636 1/20 0.34
PEPD P12955 1/20 0.34
ALOX15 P16050 1/20 0.34
PTGS1 P23219 1/20 0.34
HTR2A P28223 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL522330 0.81 NPSR1 (0.44) NPSR1ALDH1A1L3MBTL1ACE
SCHEMBL522331 0.81 NPSR1 (0.44) NPSR1ALDH1A1L3MBTL1ACE
SCHEMBL523208 0.81 NPSR1 (0.44) NPSR1ALDH1A1L3MBTL1ACE
SCHEMBL523723 0.74 EGLN1 (0.46) ALDH1A1ACEOPRM1OPRD1OPRK1
SCHEMBL523649 0.74 EGLN1 (0.46) ALDH1A1ACEOPRM1OPRD1OPRK1
SCHEMBL523650 0.74 EGLN1 (0.46) ALDH1A1ACEOPRM1OPRD1OPRK1
SCHEMBL1030669 0.69 EGLN1 (0.36) KDM4ELMNA
SCHEMBL1028657 0.69 EGLN1 (0.36) KDM4ELMNA
SCHEMBL2040068 0.66 TSHR (0.47) NPSR1ALDH1A1L3MBTL1
SCHEMBL24728099 0.65 ALDH1A1 (0.69) NPSR1ALDH1A1L3MBTL1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009002533-A1 INFLAMMATORY BOWEL DISEASE THERAPIES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2008-12-31 WO disclosed