SCHEMBL4757204

SCHEMBL4757204

Cc1cc(F)c(C(=O)Nc2ncc(S(C)(=O)=O)s2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 1/20 0.44
GRM4 Q14833 5/20 0.42
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
SCN9A Q15858 9/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
AHR P35869 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757200 0.90 FFAR2 (0.47) FFAR2GRM4CRHBPCRHR2KDM4E
SCHEMBL10114545 0.84 SCN9A (0.41) FFAR2GRM4SCN9ASMN1; SMN2NPC1
SCHEMBL4756947 0.83 FFAR2 (0.47) FFAR2GRM4CRHBPCRHR2SCN9A
SCHEMBL4756645 0.83 NPC1 (0.41) FFAR2GRM4CRHBPCRHR2SMN1; SMN2
SCHEMBL4757189 0.79 FFAR2 (0.48) FFAR2GRM4SMN1; SMN2KDM4ERXFP1
SCHEMBL4757308 0.77 KDM4E (0.41) SMN1; SMN2KDM4ERXFP1NPC1RAB9A
SCHEMBL4756975 0.77 FFAR2 (0.48) FFAR2GRM4CRHBPCRHR2SMN1; SMN2
SCHEMBL4756965 0.77 FFAR2 (0.48) FFAR2GRM4CRHBPCRHR2SMN1; SMN2
SCHEMBL4757157 0.76 STAT3 (0.49) FFAR2CRHBPCRHR2SMN1; SMN2KDM4E
SCHEMBL10114566 0.76 ALDH1A1 (0.45) FFAR2GRM4CRHBPCRHR2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES, L.C. 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC FFAR2 4045/4885GRM4 4380/4885CRHBP 3994/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.