SCHEMBL4757414

SCHEMBL4757414

O=C1OCCNC1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.47
SLC22A1 O15245 1/20 0.47
PRCP P42785 1/20 0.47
GHSR Q92847 8/20 0.46
CACNA1G O43497 2/20 0.46
ADRB2 P07550 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664410 0.83 HDAC8 (0.54) HDAC8SLC22A1PRCPCACNA1G
SCHEMBL27386827 0.77 SLC22A1 (0.60) HDAC8SLC22A1PRCPADRB2
SCHEMBL14615969 0.77 SLC22A1 (0.60) HDAC8SLC22A1PRCPADRB2
SCHEMBL2564483 0.75 PARP1 (0.37) GHSR
SCHEMBL9142562 0.73 CYP3A4 (0.49) HDAC8CACNA1G
SCHEMBL9437533 0.72 GLA (0.58) HDAC8SLC22A1PRCPGHSRADRB2
SCHEMBL9437531 0.72 GLA (0.58) HDAC8SLC22A1PRCPGHSRADRB2
SCHEMBL6936657 0.72 GLA (0.58) HDAC8SLC22A1PRCPGHSRADRB2
SCHEMBL12534333 0.72
SCHEMBL9051041 0.72 SLC6A2 (0.44) PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001203-A2 AN IMPROVED PROCESS FOR THE PREPARATION OF APREPITANT ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2008-12-31 WO disclosed