SCHEMBL4757713

SCHEMBL4757713

COC(=O)c1sc(-c2ccc(-c3cc4ncccn4n3)s2)cc1N(CC(F)(F)F)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
HTT P42858 1/20 0.32
ATM Q13315 1/20 0.32
CYP2E1 P05181 1/20 0.31
JAK2 O60674 2/20 0.31
JAK3 P52333 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828339 0.93 KDM4E (0.36) KDM4EHTTATMCYP2E1JAK2
SCHEMBL4828338 0.93 KDM4E (0.36) KDM4EHTTATMCYP2E1JAK2
SCHEMBL4789892 0.93 CYP2E1 (0.36) CYP2E1JAK2JAK3
SCHEMBL4755689 0.90 KDM4E (0.32) KDM4EHTTATMCYP2E1
SCHEMBL4823086 0.86 CYP2E1 (0.36) CYP2E1JAK2JAK3
SCHEMBL4823092 0.86 CYP2E1 (0.36) CYP2E1JAK2JAK3
Ammonia Solution, Strong SCHEMBL4819230 0.85 CYP2E1 (0.36) CYP2E1JAK2JAK3
Ammonia Solution, Strong SCHEMBL4819219 0.85 CYP2E1 (0.36) CYP2E1JAK2JAK3
SCHEMBL4143061 0.85 KDM4E (0.33) KDM4EHTTATM
SCHEMBL4155397 0.84 KDM4E (0.38) KDM4EHTTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed