SCHEMBL4789892

SCHEMBL4789892

C[C@H]1CC[C@H](C(=O)N(CC(F)(F)F)c2cc(-c3ccc(-c4cc5ncccn5n4)s3)sc2C(=O)O)CC1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.36
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
NR1I2 O75469 2/20 0.32
JAK2 O60674 2/20 0.32
JAK3 P52333 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757713 0.93 KDM4E (0.32) CYP2E1JAK2JAK3
SCHEMBL4823086 0.92 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GNR1I2JAK2
SCHEMBL4823092 0.92 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GNR1I2JAK2
Ammonia Solution, Strong SCHEMBL4819219 0.92 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GNR1I2JAK2
Ammonia Solution, Strong SCHEMBL4819230 0.92 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GNR1I2JAK2
SCHEMBL4815926 0.89 CYP2E1 (0.36) CYP2E1APOBEC3AAPOBEC3GNR1I2
SCHEMBL4828338 0.87 KDM4E (0.36) CYP2E1JAK2JAK3
SCHEMBL4828339 0.87 KDM4E (0.36) CYP2E1JAK2JAK3
SCHEMBL4157936 0.84 APOBEC3A (0.35) CYP2E1APOBEC3AAPOBEC3GNR1I2
SCHEMBL4755689 0.83 KDM4E (0.32) CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO claimed
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed
WO-2009000818-A1 3-CARBONYLAMINOTHIOPHENE-2-CARBOXYLIC ACIDS AS HEPATITIS C VIRUS INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-31 WO disclosed