SCHEMBL4758388

SCHEMBL4758388

Cc1cc(Br)cc(C)c1CC=CCNc1cccc(C(CC(=O)O)NC(=O)OCc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.41
CTSK P43235 1/20 0.39
CASP1 P29466 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8242486 0.81 PPARG (0.42) PPARG
SCHEMBL13619509 0.81 PPARG (0.42) PPARG
SCHEMBL3857652 0.77 PPARG (0.45) PPARG
SCHEMBL7061672 0.73 PPARG (0.51) PPARG
SCHEMBL6955527 0.72 CASP1 (0.60) CASP1
SCHEMBL6156731 0.72 CASP1 (0.60) CASP1
SCHEMBL6156740 0.72 CASP1 (0.60) CASP1
SCHEMBL4359028 0.72 PPARG (0.41) PPARG
SCHEMBL4359031 0.72 PPARG (0.41) PPARG
SCHEMBL4359035 0.72 PPARG (0.41) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1971582-A1 MACROCYCLIC FACTOR VIIA INHIBITORS USEFUL AS ANTICOAGULANTS Brystol-Myers Squibb Company (US) 2008-09-24 EP disclosed
WO-2007076431-A1 MACROCYCLIC FACTOR VIIA INHIBITORS USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-05 WO disclosed