SCHEMBL4758611

SCHEMBL4758611

Cc1ccccc1C(=O)OC(C)COC(=O)N[C@H](CO)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.44
ADRB2 P07550 2/20 0.44
ADRB1 P08588 2/20 0.44
ADRB3 P13945 2/20 0.44
KDM4E B2RXH2 1/20 0.43
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 1/20 0.37
PDCD1 Q15116 3/20 0.37
CD274 Q9NZQ7 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CTSS P25774 2/20 0.35
UTS2R Q9UKP6 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3106415 0.84 SMN1; SMN2 (0.41) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL4402023 0.83 ADRB2 (0.44) SMN1; SMN2ADRB2ADRB1ADRB3SCN1A
SCHEMBL3106421 0.83 ADRB2 (0.44) SMN1; SMN2ADRB2ADRB1ADRB3SCN1A
SCHEMBL4758614 0.81 TSHR (0.43) SMN1; SMN2ADRB2ADRB1ADRB3SCN1A
SCHEMBL17797889 0.79 ALDH1A1 (0.62) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL15110945 0.77 SMN1; SMN2 (0.58) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL17797803 0.75 ALDH1A1 (0.55) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL29674421 0.75 ALDH1A1 (0.55) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL17797818 0.75 ALDH1A1 (0.55) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E
SCHEMBL16048344 0.75 ALDH1A1 (0.55) SMN1; SMN2ADRB2ADRB1ADRB3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008013860-A2 ACYLOXYALKYL CARBAMATE PRODRUGS OF ALPHA-AMINO ACIDS, METHODS OF SYNTHESIS AND USE XENOPORT, INC. (US) 2008-01-31 WO claimed
WO-2008013860-A2 ACYLOXYALKYL CARBAMATE PRODRUGS OF ALPHA-AMINO ACIDS, METHODS OF SYNTHESIS AND USE XENOPORT, INC. (US) 2008-01-31 WO disclosed