SCHEMBL4758708

SCHEMBL4758708

C=CC(=O)N1C[C@H](COC(=O)N[C@H](C)c2cccc3ccccc23)[C@@H](c2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 3/20 0.41
CASR P41180 5/20 0.39
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
CCR5 P51681 1/20 0.38
EPHX2 P34913 2/20 0.38
CYP2D6 P10635 2/20 0.38
TGM2 P21980 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105648 0.78 CCR5 (0.40) CASRCCR5CYP2D6
SCHEMBL4758707 0.75 CCR5 (0.39) CCR5
SCHEMBL4100917 0.73 CASR (0.47) CASR
SCHEMBL4104683 0.73 CASR (0.50) CASRCCR5CYP2D6
SCHEMBL3573546 0.73 CASR (0.39) SSTR4CASRCYP2D6
SCHEMBL4102217 0.73 CASR (0.49) CASRCCR5CYP2D6
SCHEMBL4099302 0.72 CASR (0.47) CASRCYP2D6
SCHEMBL4099293 0.72 CASR (0.47) CASRCYP2D6
Hydrochloric Acid SCHEMBL4100877 0.72 CASR (0.49) CASR
Hydrochloric Acid SCHEMBL4106149 0.72 CASR (0.49) CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882684-A1 PYRROLIDINE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2008-01-30 EP disclosed