SCHEMBL4758707

SCHEMBL4758707

C=CC(=O)N1C[C@H](CC[C@@H](OC(N)=O)c2cccc3ccccc23)[C@@H](c2ccccc2)C1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.39
ACHE P22303 1/20 0.37
KRAS P01116 3/20 0.34
RORC P51449 3/20 0.34
BTK Q06187 3/20 0.33
TEAD1 P28347 1/20 0.33
TEAD3 Q99594 1/20 0.33
LCK P06239 1/20 0.33
SRC P12931 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105648 0.76 CCR5 (0.40) CCR5ACHEKRASRORC
SCHEMBL4758705 0.76 CCR5 (0.39) CCR5ACHEKRASRORCTEAD1
SCHEMBL4758708 0.75 SSTR4 (0.41) CCR5
SCHEMBL3573544 0.71 AOC3 (0.33) CCR5
SCHEMBL11566786 0.71 AOC3 (0.46) ALDH1A1
SCHEMBL4108113 0.69 CCR5 (0.42) CCR5RORC
SCHEMBL4108109 0.69 CCR5 (0.42) CCR5RORC
SCHEMBL7187735 0.67 HPGD (0.52) ALDH1A1
SCHEMBL8038236 0.66 AOC3 (0.40)
SCHEMBL11567917 0.66 KDM4E (0.49) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882684-A1 PYRROLIDINE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2008-01-30 EP disclosed