SCHEMBL4759340

SCHEMBL4759340

O=C(NCc1c[nH]cn1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
LMNA P02545 2/20 0.51
POLB P06746 1/20 0.51
RAB9A P51151 1/20 0.51
HPGD P15428 3/20 0.49
KDM4E B2RXH2 2/20 0.49
GAA P10253 1/20 0.49
MAPK14 Q16539 1/20 0.48
HDAC6 Q9UBN7 3/20 0.46
HDAC1 Q13547 2/20 0.46
ALDH1A1 P00352 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
MIF P14174 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
ERCC1 P07992 1/20 0.44
ERCC4 Q92889 1/20 0.44
PRSS1 P07477 1/20 0.44
CTSG P08311 1/20 0.44
CTRB1 P17538 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17548986 0.89 HDAC2 (0.47) NPC1LMNAPOLBRAB9AKDM4E
SCHEMBL6972274 0.86 HDAC6 (0.55) POLBKDM4EHDAC6HDAC1L3MBTL1
SCHEMBL1300262 0.85 MAPT (0.52) NPC1LMNAPOLBRAB9AHPGD
SCHEMBL13213701 0.85 KDM4E (0.47) NPC1LMNAPOLBRAB9AHPGD
SCHEMBL1300005 0.82 GAA (0.44) NPC1LMNAPOLBRAB9AHPGD
SCHEMBL6973879 0.82 HDAC6 (0.54) LMNAPOLBRAB9AHPGDKDM4E
SCHEMBL20501735 0.80 SMN1; SMN2 (0.34) NPC1LMNAPOLBRAB9AHPGD
SCHEMBL28255183 0.79 TSHR (0.54) NPC1POLBRAB9AGAAKMT2A
SCHEMBL21820359 0.76 RAB9A (0.46) NPC1POLBRAB9AGAAHDAC6
SCHEMBL1310658 0.76 ACE (0.48) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928879-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS Brystol-Myers Squibb Company (US) 2008-06-11 EP claimed
WO-2007038314-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-04-05 WO claimed