SCHEMBL4759730

SCHEMBL4759730

COc1cc(C(=O)[C@H]2C(=O)c3cc(-c4noc(=O)[nH]4)ccc3OC23CCNCC3)nc2c(OC)cccc12

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TNKS O95271 10/20 0.34
TNKS2 Q9H2K2 10/20 0.34
PARP1 P09874 5/20 0.34
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
PARP2 Q9UGN5 6/20 0.33
PTGER4 P35408 1/20 0.32
AGTR1 P30556 1/20 0.32
JUND P17535 1/20 0.32
FOSB P53539 1/20 0.32
XIAP P98170 1/20 0.32
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759789 0.89 TNKS (0.34) TNKSTNKS2PARP1ACACBACACA
SCHEMBL4412678 0.87 ACACB (0.35) TNKSTNKS2PARP1ACACBACACA
SCHEMBL2362040 0.87 ACACB (0.35) TNKSTNKS2PARP1ACACBACACA
SCHEMBL4708996 0.87 ACACA (0.35) TNKSTNKS2PARP1ACACBACACA
SCHEMBL4760383 0.86 ACACB (0.34) TNKSTNKS2PARP1ACACBACACA
SCHEMBL4760480 0.85 NOTUM (0.36) ACACBACACAPTGER4
SCHEMBL4708583 0.85 XIAP (0.39) TNKSTNKS2ACACBACACAPARP2
SCHEMBL4760214 0.85 ACACA (0.34) TNKSTNKS2PARP1ACACBACACA
SCHEMBL4707267 0.84 ACACA (0.38) TNKSTNKS2ACACBACACAPARP2
SCHEMBL4711163 0.84 ACACA (0.34) TNKSTNKS2PARP1ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP claimed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO claimed
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP disclosed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed