SCHEMBL4759913

SCHEMBL4759913

CC(C)CC(C(=O)NC1(C#N)CC1)c1cccc(-c2cccc(-c3csc(N4CCNCC4)n3)c2)c1

nearest known ligand 0.78

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.78
CTSS P25774 19/20 0.78
CTSL P07711 18/20 0.78
CTSB P07858 16/20 0.78
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760512 0.96 CTSK (0.78) CTSKCTSSCTSLCTSBKCNH2
SCHEMBL4790513 0.92 CTSK (0.78) CTSKCTSSCTSLCTSBKCNH2
SCHEMBL4760896 0.88 CTSK (0.72) CTSKCTSSCTSLCTSBKCNH2
SCHEMBL4716426 0.88 CTSK (1.00) CTSKCTSSCTSLCTSB
SCHEMBL4717266 0.84 CTSK (0.79) CTSKCTSSCTSLCTSB
SCHEMBL4714257 0.84 CTSL (1.00) CTSKCTSSCTSLCTSB
SCHEMBL4761353 0.83 CTSK (1.00) CTSKCTSSCTSLCTSB
SCHEMBL6183387 0.80 CTSK (0.60) CTSKCTSSCTSLCTSB
SCHEMBL7606091 0.80 CTSK (0.60) CTSKCTSSCTSLCTSB
SCHEMBL4713651 0.80 CTSK (0.79) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1248612-B1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-02-27 EP claimed