SCHEMBL4760263

SCHEMBL4760263

O=C1CSc2cc(F)c(OC(=O)O)cc2N1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
MAOA P21397 6/20 0.44
MAOB P27338 6/20 0.44
KMT2A Q03164 2/20 0.41
EPHX2 P34913 1/20 0.41
HPGD P15428 1/20 0.40
TRPV1 Q8NER1 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760038 0.83 KMT2A (0.48) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL3063917 0.78 HTT (0.57) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL3069824 0.73 MAOB (0.49) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL7451837 0.72 MAOA (0.47) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL14341235 0.72 EPHX2 (0.56) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL1223787 0.72 MAOA (0.47) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL30954132 0.72 MAOA (0.47) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL5748824 0.70 HTT (0.46) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL3077002 0.70 KMT2A (0.49) HTTALDH1A1LMNAMAOAMAOB
SCHEMBL13014026 0.69 KMT2A (0.60) HTTALDH1A1LMNAMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943222-A1 ANTIBACTERIAL ACTIVE 5-CHINOLIN DERIVATIVE Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2008-07-16 EP disclosed
WO-2007042325-A1 ANTIBACTERIAL ACTIVE 5-CHINOLIN DERIVATIVE Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2007-04-19 WO disclosed