SCHEMBL4760703

SCHEMBL4760703

c1ccc2nc(-n3ccnn3)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 6/20 0.44
HRH3 Q9Y5N1 5/20 0.44
KDM4E B2RXH2 4/20 0.44
CYP1A2 P05177 3/20 0.44
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
USP2 O75604 1/20 0.44
ADRB1 P08588 1/20 0.44
CYP3A4 P08684 1/20 0.44
HTR1A P08908 1/20 0.44
HTR2C P28335 1/20 0.44
MAPK1 P28482 1/20 0.44
SLC6A4 P31645 1/20 0.44
HTR7 P34969 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5279937 0.98 NPC1 (0.44) NPC1RAB9AALDH1A1HRH3KDM4E
SCHEMBL30344655 0.76 ALDH1A1 (0.48) NPC1RAB9AALDH1A1HRH3KDM4E
SCHEMBL3806773 0.76 ALDH1A1 (0.48) NPC1RAB9AALDH1A1HRH3KDM4E
SCHEMBL10609919 0.75 ALDH1A1 (0.49) NPC1RAB9AALDH1A1HRH3KDM4E
SCHEMBL27926914 0.75 LMNA (0.52) ALDH1A1KDM4ETDP1CYP3A4HTR2C
SCHEMBL4760702 0.73 NOTUM (0.40) ALDH1A1KDM4ETDP1HSD17B10MAP3K5
SCHEMBL4448982 0.73 GAA (0.49) NPC1RAB9AALDH1A1KDM4ECYP1A2
Hydrochloric Acid SCHEMBL5279933 0.72 NOTUM (0.39) RAB9AALDH1A1KDM4ETDP1HTT
SCHEMBL24240280 0.72 NOTUM (0.48) CYP1A2HTR3AMAP3K5NOTUM
Quinoline SCHEMBL27588058 0.71 ALDH1A1 (0.55) NPC1RAB9AALDH1A1KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917013-A1 USE OF AZABICYCLO HEXANE DERIVATIVES GLAXO GROUP LIMITED (GB) 2008-05-07 EP disclosed
WO-2007022980-A1 USE OF AZABICYCLO HEXANE DERIVATIVES GLAXO GROUP LIMITED (GB) 2007-03-01 WO disclosed