SCHEMBL4760914

SCHEMBL4760914

C[C@]1(COc2ccccc2C#N)CO1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPK1 P28482 1/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
MAOA P21397 1/20 0.41
HTR2B P41595 1/20 0.41
GAA P10253 2/20 0.41
POLB P06746 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM4E B2RXH2 2/20 0.39
TP53 P04637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3153812 1.00 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL19527776 0.83 DHFR (0.46) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL3154239 0.82 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL3149891 0.79 ALDH1A1 (0.33) ALDH1A1MAPK1HPGDNPC1RAB9A
SCHEMBL3149885 0.79 ALDH1A1 (0.33) ALDH1A1MAPK1HPGDNPC1RAB9A
SCHEMBL30079702 0.77 SMN1; SMN2 (0.42) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL4451541 0.77 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL10887533 0.76 POLB (0.44) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL19612210 0.75 IDO1 (0.36) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR
SCHEMBL19527479 0.75 TP53 (0.41) ALDH1A1SMN1; SMN2MAPK1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945613-A1 NOVEL 1 -BENZYL-4-PIPERIDINAMINES THAT ARE USEFUL IN THE TREATMENT OF COPD AND ASTHMA AstraZeneca AB (SE) 2008-07-23 EP disclosed
WO-2007053082-A1 NOVEL 1 -BENZYL-4-PIPERIDINAMINES THAT ARE USEFUL IN THE TREATMENT OF COPD AND ASTHMA ASTRAZENECA AB (SE) 2007-05-10 WO disclosed