SCHEMBL4760926

SCHEMBL4760926

CC1(C)CCC(C)(C)c2cc(Cn3cccn3)c(CCc3ccc(O)cc3)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 2/20 0.40
TSHR P16473 2/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPT P10636 3/20 0.37
GAA P10253 2/20 0.37
BRD4 O60885 1/20 0.37
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CYP26A1 O43174 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22163720 0.87 RXRA (0.50) HTTHDAC1HDAC6
SCHEMBL4709673 0.83 MEN1 (0.39) KMT2AMEN1ALDH1A1HTTTSHR
SCHEMBL4710162 0.82 HTT (0.43) KMT2AMEN1ALDH1A1HTTMAPT
SCHEMBL4710160 0.80 AGTR1 (0.42) KMT2AMEN1ALDH1A1HTTCYP2C9
SCHEMBL4710917 0.78 LPAR1 (0.41) KMT2AMEN1ALDH1A1HTTTSHR
SCHEMBL4710916 0.78 HTT (0.39) KMT2AMEN1ALDH1A1HTTTSHR
SCHEMBL4709265 0.75 BRD4 (0.37) KMT2AMEN1ALDH1A1HTTTSHR
SCHEMBL14159946 0.74 CYP26A1 (0.47) HTTCYP26A1CYP26B1
SCHEMBL14159944 0.72 CYP3A4 (0.48) KMT2AMEN1HTTHDAC1HDAC6
SCHEMBL4711568 0.72 MEN1 (0.35) KMT2AMEN1ALDH1A1HTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1935869-A1 Retinoids for the treatment of emphysema F. HOFFMANN-LA ROCHE AG (CH) 2008-06-25 EP disclosed