SCHEMBL4763203

SCHEMBL4763203

CN(C)c1ccc(Nc2ncc3c(=O)c(C(=O)O)cn(C4CCCCC4)c3n2)cc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 7/20 0.62
CCNT1 O60563 1/20 0.47
CDK9 P50750 1/20 0.47
AURKA O14965 5/20 0.46
CDK1 P06493 4/20 0.46
CCNB1 P14635 4/20 0.46
SYK P43405 1/20 0.46
CDK4 P11802 4/20 0.44
CCND1 P24385 4/20 0.44
KDM4E B2RXH2 1/20 0.44
CCND2 P30279 2/20 0.44
CCND3 P30281 2/20 0.44
WEE1 P30291 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527782 0.88 CSF1R (0.57) CSF1RCCNT1CDK9AURKACDK1
SCHEMBL4767401 0.84 CSF1R (0.86) CSF1RAURKACDK1CCNB1CDK4
SCHEMBL4884345 0.84 CSF1R (0.81) CSF1RAURKACDK1CDK4WEE1
SCHEMBL4889961 0.84 CSF1R (0.60) CSF1RCCNT1CDK9AURKACDK1
SCHEMBL4791572 0.83 CSF1R (0.86) CSF1RAURKACDK1CCNB1CDK4
SCHEMBL4891427 0.83 CSF1R (0.60) CSF1RAURKACDK1SYKCDK4
SCHEMBL4891439 0.83 CSF1R (0.69) CSF1RSYKCDK4CCND1CCND2
SCHEMBL4890824 0.83 CSF1R (0.66) CSF1RCCNT1CDK9CDK4CCND1
SCHEMBL4882532 0.82 CSF1R (0.80) CSF1R
SCHEMBL4885531 0.82 CSF1R (0.68) CSF1RSYKCDK4CCND1CCND2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937681-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-02 EP disclosed
WO-2007033232-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO disclosed