SCHEMBL4763436

SCHEMBL4763436

O=C(NC1=COCO1)c1cc[nH]c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R8 Q9NYW2 1/20 0.35
NPC1 O15118 7/20 0.33
RAB9A P51151 7/20 0.33
SMN1; SMN2 Q16637 5/20 0.33
PKM P14618 2/20 0.33
CASP3 P42574 5/20 0.32
SENP7 Q9BQF6 5/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
TP53 P04637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PTGS2 P35354 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31228747 0.69 PTPN1 (0.58) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6954756 0.69 PTPN1 (0.58) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6246004 0.68
SCHEMBL6037520 0.67 RAB9A (0.67) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL8772217 0.67 POLB (0.54) NPC1RAB9ASMN1; SMN2PKMMEN1
SCHEMBL18993451 0.67 NPC1 (0.43) TAS2R8NPC1RAB9ASMN1; SMN2PKM
SCHEMBL6037515 0.67 NPC1 (0.43) TAS2R8NPC1RAB9ASMN1; SMN2PKM
SCHEMBL16416801 0.67 KDM4E (0.67) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6224947 0.66
SCHEMBL1072537 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004623-A1 PYRIDYL- AND PYRIMIDINYL-SUBSTITUTED PYRROLE-, THIOPHENE- AND FURANE-DERIVATIVES AS KINASE INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2008-12-24 EP disclosed
WO-2007110344-A1 PYRIDYL- AND PYRIMIDINYL-SUBSTITUTED PYRROLE-, THIOPHENE- AND FURANE-DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2007-10-04 WO disclosed