SCHEMBL4764579

SCHEMBL4764579

[CH2]CN1CCC(n2ccc3c(Cl)c(C)[nH]c3c2=O)CC1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.34
DRD4 P21917 7/20 0.34
DRD3 P35462 7/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
IDH1 O75874 1/20 0.31
SLC6A4 P31645 2/20 0.31
OPRM1 P35372 2/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
HTR2A P28223 1/20 0.31
SLC2A1 P11166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766195 0.85 DRD2 (0.52) DRD2DRD4DRD3OPRM1
SCHEMBL4764601 0.82 TP53 (0.33) L3MBTL1MEN1KMT2AHTR2ASLC2A1
SCHEMBL4868563 0.72 ABCC2 (0.45)
SCHEMBL4764944 0.72 SCD (0.33)
SCHEMBL4869753 0.70 HRH3 (0.33) MEN1KMT2AIDH1
SCHEMBL4873377 0.70 JAK2 (0.34) HTR2A
SCHEMBL4879836 0.70 ABCC2 (0.38)
SCHEMBL4874945 0.69 ITGAL (0.38) MEN1KMT2A
SCHEMBL12668544 0.56 CYP1A2 (0.43)
SCHEMBL16651267 0.55 KDM5A (0.44) IDH1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991545-A2 ANTIBACTERIAL PYRROLOPYRIDINES, PYRROLOPYRIMIDINES, AND PYRROLOAZEPINES AstraZeneca AB (SE) 2008-11-19 EP claimed
WO-2007071965-A2 ANTIBACTERIAL PYRROLOPYRIDINES, PYRROLOPYRIMIDINES, AND PYRROLOAZEPINES ASTRAZENECA AB (SE) 2007-06-28 WO claimed