SCHEMBL4764922

SCHEMBL4764922

O=C(O)C(F)C(=O)c1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.52
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LTA4H P09960 1/20 0.44
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
PLOD2 O00469 2/20 0.42
PLOD3 O60568 2/20 0.42
PLOD1 Q02809 2/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
HIF1A Q16665 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MPO P05164 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2A6 P11509 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5428890 0.98 NAPRT (0.50) NAPRTMEN1KMT2ALTA4HALDH1A1
SCHEMBL2851869 0.82 NAPRT (0.45) NAPRTMEN1KMT2ALTA4HALDH1A1
SCHEMBL10767862 0.80 TDP1 (0.52) NAPRTMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5141652 0.78 TDP1 (0.50) NAPRTMEN1KMT2AALDH1A1CYP3A4
SCHEMBL27566013 0.77 ALDH1A1 (0.58) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL3844697 0.75 NAPRT (0.52) NAPRTMEN1KMT2AALDH1A1CYP1A2
SCHEMBL28624819 0.75 NAPRT (0.52) NAPRTMEN1KMT2ALTA4HALDH1A1
SCHEMBL1380026 0.74 KMT2A (0.45) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL6007960 0.73 NAPRT (0.50) NAPRTMEN1KMT2ALTA4HALDH1A1
SCHEMBL6007952 0.73 NAPRT (0.50) NAPRTMEN1KMT2ALTA4HALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1674456-B1 Use of 2-fluoro- 3-ketoesters for preparing 3-fluoro-6,7,8,9-tetrahydro-4-H-pyrimdo[1,2-a]pyrimidin-4-ones SANOFI AVENTIS (FR) 2008-07-16 EP claimed
EP-1603876-B1 PROCESS FOR THE PREPARATION OF PYRIDINYL AND PYRIMIDINYL MONO-FLUORINATED BETA KETO ESTERS SANOFI AVENTIS (FR) 2007-02-14 EP claimed