SCHEMBL4765296

SCHEMBL4765296

CCCn1c(C=Cc2cnn(-c3ccccc3)c2)c([N+](=O)[O-])c(=O)n(C(C)OC)c1=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
POLB P06746 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPK1 P28482 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MITF O75030 1/20 0.34
LMNA P02545 2/20 0.34
HSP90AA1 P07900 1/20 0.33
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765284 1.00 NPC1 (0.40) NPC1RAB9AADORA2AADORA2BADORA1
SCHEMBL4766270 0.89 SMN1; SMN2 (0.41) NPC1RAB9AMAPTSMN1; SMN2POLB
SCHEMBL4766280 0.89 SMN1; SMN2 (0.41) NPC1RAB9AMAPTSMN1; SMN2POLB
SCHEMBL4763478 0.89 NCOA1 (0.42) NPC1RAB9AADORA2AADORA2BADORA1
SCHEMBL4763471 0.89 NCOA1 (0.42) NPC1RAB9AADORA2AADORA2BADORA1
SCHEMBL4771171 0.87 MAPT (0.39) MAPTSMN1; SMN2POLBNCOA1NCOA3
SCHEMBL4771156 0.87 MAPT (0.39) MAPTSMN1; SMN2POLBNCOA1NCOA3
SCHEMBL4765287 0.85 ADORA2A (0.42) NPC1RAB9AADORA2AADORA2BADORA1
SCHEMBL4770893 0.84 ADORA2A (0.45) NPC1RAB9AADORA2AADORA2BADORA1
SCHEMBL4770873 0.84 ADORA2A (0.45) NPC1RAB9AADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed