SCHEMBL4763471

SCHEMBL4763471

CCCCn1c(=O)c([N+](=O)[O-])c(/C=C/c2cnn(-c3ccccc3)c2)n(C(C)OC)c1=O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MAPT P10636 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPK1 P28482 1/20 0.38
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
MITF O75030 1/20 0.34
LMNA P02545 3/20 0.34
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763478 1.00 NCOA1 (0.42) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4765284 0.89 NPC1 (0.40) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4765296 0.89 NPC1 (0.40) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4767902 0.89 NCOA1 (0.42) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4767911 0.89 NCOA1 (0.42) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4769732 0.87 NCOA1 (0.44) NCOA1NCOA3MAPTSMN1; SMN2POLB
SCHEMBL4769724 0.87 NCOA1 (0.44) NCOA1NCOA3MAPTSMN1; SMN2POLB
SCHEMBL4766280 0.87 SMN1; SMN2 (0.41) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4766270 0.87 SMN1; SMN2 (0.41) NCOA1NCOA3NPC1RAB9AMAPT
SCHEMBL4763475 0.87 NCOA1 (0.42) NCOA1NCOA3NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed