SCHEMBL4765824

SCHEMBL4765824

CCc1cc(N)c(CC=O)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.51
P2RX3 P56373 2/20 0.39
P2RX2 Q9UBL9 2/20 0.39
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
HTR2A P28223 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP19A1 P11511 1/20 0.36
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772225 0.93 TAAR1 (0.47) TAAR1P2RX3P2RX2GAAMAPT
SCHEMBL1579468 0.87 KDM4E (0.42) TAAR1GAAMAPTTSHRMAPK1
SCHEMBL7256087 0.82 GAA (0.46) TAAR1GAAMAPTTSHRMAPK1
SCHEMBL577652 0.81 GAA (0.55) TAAR1GAAMAPTMAPK1RAB9A
SCHEMBL4768439 0.81 TAAR1 (0.39) TAAR1MAPK1HTTHTR2ARAB9A
SCHEMBL21798818 0.81 TAAR1 (0.45) TAAR1GAAMAPTTSHRMAPK1
SCHEMBL4847393 0.79 TAAR1 (0.47) TAAR1P2RX3P2RX2MAPTTSHR
SCHEMBL5951991 0.79 TAAR1 (0.59) TAAR1P2RX3P2RX2GAAMAPT
SCHEMBL27749404 0.79 ALDH1A1 (0.32)
SCHEMBL17653319 0.78 HTR2A (0.44) TAAR1MAPTHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989195-A1 PHOSPHODIESTERASE 10 INHIBITORS Amgen Inc. (US) 2008-11-12 EP disclosed
WO-2007103260-A1 PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC. (US) 2007-09-13 WO disclosed