SCHEMBL4766003

SCHEMBL4766003

CC(c1ccccc1)n1c(/C=C/c2cnn(Cc3ccccc3C(F)(F)F)c2)c([N+](=O)[O-])c(=O)n(C2CCC2)c1=O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
C5AR1 P21730 9/20 0.33
TAS2R8 Q9NYW2 1/20 0.32
HSD11B1 P28845 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPK1 P28482 1/20 0.31
GNRHR P30968 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766009 1.00 TACR1 (0.33) TACR1ADORA2AADORA2BADORA1C5AR1
SCHEMBL4763444 0.91 MAPT (0.33) ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4763440 0.91 MAPT (0.33) ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4763163 0.89 ADORA2A (0.37) ADORA2AADORA2BADORA1TAS2R8ALDH1A1
SCHEMBL4763169 0.89 ADORA2A (0.37) ADORA2AADORA2BADORA1TAS2R8ALDH1A1
SCHEMBL4762674 0.88 ADORA2A (0.36) ADORA2AADORA2BADORA1C5AR1TAS2R8
SCHEMBL4762676 0.88 ADORA2A (0.36) ADORA2AADORA2BADORA1C5AR1TAS2R8
SCHEMBL4891718 0.86 ADORA2B (0.41) TACR1ADORA2AADORA2BADORA1C5AR1
SCHEMBL4766007 0.84 C5AR1 (0.41) ADORA2AADORA2BADORA1C5AR1HSD11B1
SCHEMBL4771502 0.84 MAPT (0.35) ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed