SCHEMBL4766007

SCHEMBL4766007

O=c1c([N+](=O)[O-])c(/C=C/c2cnn(Cc3ccccc3C(F)(F)F)c2)n(CCc2ccccc2)c(=O)n1C1CCC1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 18/20 0.41
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763441 0.91 TP53 (0.34) C5AR1ADORA2AADORA2BADORA1
SCHEMBL4762674 0.90 ADORA2A (0.36) C5AR1ADORA2AADORA2BADORA1HSD11B1
SCHEMBL4762676 0.90 ADORA2A (0.36) C5AR1ADORA2AADORA2BADORA1HSD11B1
SCHEMBL4763165 0.89 ADORA2B (0.43) C5AR1ADORA2AADORA2BADORA1
SCHEMBL4763171 0.89 ADORA2B (0.43) C5AR1ADORA2AADORA2BADORA1
SCHEMBL4891723 0.86 C5AR1 (0.42) C5AR1ADORA2AADORA2BADORA1HSD11B1
SCHEMBL4769025 0.85 C5AR1 (0.37) C5AR1ADORA2AADORA2BADORA1HSD11B1
SCHEMBL4769016 0.85 C5AR1 (0.37) C5AR1ADORA2AADORA2BADORA1HSD11B1
SCHEMBL4771507 0.85 MAPT (0.36)
SCHEMBL4766003 0.84 TACR1 (0.33) C5AR1ADORA2AADORA2BADORA1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed