SCHEMBL4766969

SCHEMBL4766969

O=C1O[C@@H](Cc2ncc[nH]2)CN1c1ccc(O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 7/20 0.50
MAOA P21397 11/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAOB P27338 4/20 0.41
LMNA P02545 1/20 0.41
PTGS1 P23219 1/20 0.41
SDHA P31040 1/20 0.41
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723657 0.82 CALML3 (0.47) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL4766974 0.81 GRM2 (0.46) CALML3
SCHEMBL10062439 0.79 CALML3 (0.67) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL542031 0.79 CALML3 (0.67) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL542030 0.79 CALML3 (0.67) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL17769240 0.78 CALML3 (0.53) CALML3MAOAMAOBLMNAPTGS1
SCHEMBL17769239 0.78 CALML3 (0.53) CALML3MAOAMAOBLMNAPTGS1
SCHEMBL7004283 0.77 CALML3 (0.48) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL7840408 0.77 CALML3 (0.70) CALML3MAOACYP3A4CYP2D6MAOB
SCHEMBL10026237 0.75 CALML3 (0.50) CALML3MAOAMAOBLMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931684-A2 OXAZOLIDINONE-QUINOLONE HYBRIDS AS ANTIBACTERIAL COMPOUNDS Actelion Pharmaceuticals Ltd. (CH) 2008-06-18 EP disclosed
WO-2007017828-A2 OXAZOLIDINONE-QUINOLONE HYBRIDS AS ANTIBACTERIAL COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2007-02-15 WO disclosed